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Drug Name: Enzastaurin Hydrochloride [USAN] View Structure
Description: A protein kinase Cbeta-selective inhibitor.

NCI: The hydrochloride salt of enzastaurin, a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, enzastaurin selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden. ... (NCI Thesaurus) 



 
 
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